Azélastine
- Azélastine
-
| Azélastine |
 |
| Énantiomère R de l'azélastine (à gauche) et S-azélastine (à droite) |
| Général |
| Nom IUPAC |
(RS)-4-[(4-chlorophényl)méthyl]-2- (1-méthylazepan-4-yl)-phtalazin-1-one |
| No CAS |
58581-89-8 |
| Code ATC |
R01AC03, R06AX19, GX07 |
| SMILES |
C1C[C@@H](CCC[N@@]1C)n1nc(c2ccccc2c1=O)Cc1ccc(cc1)Cl
PubChem, Vue 3D
|
| InChI |
InChI : Vue 3D
InChI=1/C22H24ClN3O/c1-25-13-4-5-18(12-14-25)26-22(27)20-7-3-2-6-19(20)21(24-26)15-16-8-10-17(23)11-9-16/h2-3,6-11,18H,4-5,12-15H2,1H3
|
| Propriétés chimiques |
| Formule brute |
C22H24ClN3O [Isomères]
|
| Masse molaire[1] |
381,898 ± 0,022 g·mol-1
C 69,19 %, H 6,33 %, Cl 9,28 %, N 11 %, O 4,19 %,
|
|
Unités du SI & CNTP, sauf indication contraire.
|
L'azélastine est un substance chimique médicament de la famille des phtallazinone qui possède des propriétés antihistaminiques H1 et bronchodilatatrices. C'est une molécule utilisée dans le traitement de l'allergie et de l'asthme. Il est commercialisé en France avec la spécialité Allergodil .
Voir aussi
Article connexe
Liens externes
Notes et références
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Contenu soumis à la licence CC-BY-SA. Source : Article Azélastine de Wikipédia en français (auteurs)
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